Exemestane is a very powerful aromatase inhibitor or (Ai). Originally this anti estrogen produced by Pharmacia & UpJohn was designed for use in the medical field. Exemestane would be used as a treatment option for women with breast cancer.
Exemestane was approved by the FDA as a prescription medication for breast cancer treatment back in 1999. Today, this anti estrogen drug is used in treating breast cancer patients all over the world.
Exemestane is known to lower estrogen levels in breast cancer patients by as much as 85 percent. This anti estrogen medication is usually prescribed in breast cancer treatment after first-line or initial treatment options are unsuccessful.
As a matter of fact, Exemestane will permanently restrict and completely disarm aromatase enzymes. It is this aromatase enzyme that changes anabolic steroid compounds like synthetic testosterone to estrogen. Exemestane will render the aromatase enzyme impotent and totally ineffective.
One of the benefits of Exemestane to bodybuilding is that it will hinder the level of estrogen in the body. This is particularly important to male bodybuilders who want to reap the gains of androgenic-anabolic steroid use without encountering unfavorable side effects in the process.
High estrogen levels in male bodybuilders can be detrimental to bodybuilding gains. High levels of estrogen leads to feminization effects. The classic feminization effects that most bodybuilders experience is the development of male boobs. This is a condition described in medical terms as gynecomastia.
Gynecomastia is a condition characterised by the enlargement of male breasts. Male bodybuilders are wary of this side effect which is caused by exceedingly high estrogen levels in the body.
Since testosterone converts to estrogen and many androgenic-anabolic steroids are derivatives of testosterone, the risk of bodybuilders having high estrogen levels when using anabolic steroids is great.
Another estrogen-related side effect that adversely affects male bodybuilders is water retention. Bodybuilders training hard to achieve lean, vascular muscles would be disappointed when they have full, blubby muscle mass due to the retention of water.
High estrogen levels can also slow down metabolism, leading to increased body fat and weight gain. It is important that bodybuilders engage in proper post-cycle therapy practices. Post-cycle therapy involves the use of anti estrogen drugs like Exemestane to help regulate estrogen levels while also promoting normalcy in testosterone levels.
The primary bodybuilding benefit of Exemestane lies in the drug’s aromatase inhibiting capabilities. However, using Exemestane will help bodybuilders in the following ways:
- Reduced Estrogen Levels: As an aromatase inhibitor, Exemestane will prevent the aromatase enzyme from binding with steroid compounds used. When this happens, the steroid compounds are prevented from turning into estrogen.
- Resumption of Testosterone Production: The use of Exemestane during post-cycle therapy will not only reduce estrogen levels, but also promote the resumption of testosterone production.
- Prevention of Feminization Side Effects: Exemestane will greatly reduce the occurrence of feminization side effects in male bodybuilders. This anti estrogen drug will prevent male bodybuilders from experiencing side effects like water retention, testicular atrophy, and gynecomastia.